AKR1C3-IN-5

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AKR1C3-IN-5

本产品不向个人销售，仅用作科学研究，不用于任何人体实验及非科研性质的动物实验。

包装与价格：

包装	价格(元)
100mg	电议
250mg	电议
500mg	电议

产品介绍

AKR1C3-IN-5 (Compound 6e) 是一种有效的AKR1C3抑制剂。AKR1C3 酶在激素依赖性前列腺和乳腺肿瘤中过度表达。 AKR1C3-IN-5 源自 drupanin，其对 MCF-7 细胞的半数抑制浓度 (IC₅₀) 为 9.6 ± 3 μM，选择性指数 (SI) 为 5.5。

生物活性	AKR1C3-IN-5 (Compound 6e) is a potent inhibitor ofAKR1C3. AKR1C3 enzyme is overexpressed in hormone-dependent prostate and breast tumors. AKR1C3-IN-5 derived from drupanin, which exhibits half-maximal inhibitory concentration (IC₅₀) of 9.6 ± 3 μM and selectivity index (SI) of 5.5 against MCF-7 cells^[1].
分子量	592.72
Formula	C₃₄H₄₄N₂O₇
运输条件	Room temperature in continental US; may vary elsewhere.
储存方式	Please store the product under the recommended conditions in the Certificate of Analysis.