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Cetrorelix diacetate
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Cetrorelix diacetate图片
CAS NO:130143-01-0
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品名称
SB-75 diacetate
产品介绍
Cetrorelix diacetate (SB-075 diacetate)是GnRH受体的强效拮抗剂,其IC50值为 1.21 nM。
生物活性

Cetrorelix diacetate (SB-075 diacetate) is a potent gonadotropin-releasing hormone(GnRH)receptor antagonist with anIC50of 1.21 nM[1].

IC50& Target

IC50: 1.21 nM GnRH[1].

体外研究
(In Vitro)

Cetrorelix diacetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix diacetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells[2].

Clinical Trial
分子量

1551.14

Formula

C74H100ClN17O18

CAS 号

130143-01-0

Sequence Shortening

Ac-{2-Naph-Ala}-{Cl-Phe}-{3Py-Ala}-SY-{Cit}-LRPA-NH2

中文名称

二醋酸西曲瑞克

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.