PF-4136309 racemate (INCB8761; INCB-8761; PF4136309; PF-4136309), the racemic mixture of PF-4136309, is an orally bioavailable CCR2 (C-C Motif Chemokine Receptor 2) antagonist with anticancer activity. It inhibits CCR2 with IC50 values of 5.2 nM, 17 nM and 13 nM for human, mouse and rat CCR2, respectively.

纯度：≥98%

CAS：857679-55-1