[(pF)Phe4]Nociceptin(1-13)NH2 是一种高效的选择性 NOP 受体 (OP4) 激动剂,pKi 为 10.68,pEC50 为 9.31。
Cas No. | 380620-88-2 |
化学名 | (S,Z)-6-amino-N-((S,Z)-1-(((S,Z)-1-(((S,Z)-1-(((S)-6-amino-1-hydroxy-1-iminohexan-2-yl)imino)-5-guanidino-1-hydroxypentan-2-yl)imino)-1-hydroxypropan-2-yl)imino)-1,3-dihydroxypropan-2-yl)-2-((Z)-((2S,3Z,5S,6Z,9Z,11S,12Z,14S,15Z,18Z,21Z,23S)-23-amino-2-(3- |
Canonical SMILES | C[C@@](/N=C(O)/C/N=C(O)/[C@](/N=C(O)/[C@](/N=C(O)/C/N=C(O)/C/N=C(O)/[C@](N)([H])CC1=CC=CC=C1)([H])CC2=C(F)C(F)=C(F)C(F)=C2F)([H])[C@@](O)([H])C)([H])/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](C(O)=N)([H])CCCCN)([H] |
分子式 | C61H95F5N22O15 |
分子量 | 1471.54 |
溶解度 | Soluble to 2 mg/ml in Water |
储存条件 | Desiccate at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |