LJ-4517 是一种有效的A2AAR拮抗剂，其Ki为 18.3 nM。LJ-4517 可以有效地取代 WT A2AAR 处 [3H]ZM241385 (HY-19532) 的结合。
| 生物活性 | LJ-4517 is a potentA2AARantagonist, with aKiof 18.3 nM. LJ-4517 is potent in displacing the binding of [3H]ZM241385(HY-19532) at WT A2AAR[1]. |
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体外研究
(In Vitro) | LJ-4517 (10 μM) induces cAMP accumulation[1].
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| 运输条件 | Room temperature in continental US; may vary elsewhere. |
| 储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |
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