CAS NO: | 167011-22-5 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | CP-96021 hydrochloride is a balanced, combined, potent and orally activeleukotriene D4 (LTD4)/platelet activating factor (PAF)receptor antagonist withKivalues of 34 nM and 37 nM, respectively[1]. | ||
IC50& Target[1] |
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体内研究 (In Vivo) | In vivo, CP-96021 inhibits iv LTD4- and iv PAF-induced bronchoconstriction in guinea pigs withED50s of 0.46 and 0.16 mg/kg p.o. respectively. CP-96021 effectively blocks the combined airway obstructive effects of endogenously released PAF and LTD4 stimulated by aerosolized antigen challenge in guinea pigs with anED50s of 1.8 mg/kg p.o[1]. | ||
分子量 | 529.03 | ||
Formula | C29H22ClFN4OS | ||
CAS 号 | 167011-22-5 | ||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |