CAS NO: | 139401-45-9 |
包装 | 价格(元) |
100mg | 电议 |
250mg | 电议 |
500mg | 电议 |
生物活性 | CP-96486 is a potent and orally active leukotriene D4(LTD4)/platelet activating factor (PAF) receptor antagonist withKis of 20 and 24 nM, respectively. | ||
IC50& Target |
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体外研究 (In Vitro) | CP-96486 (CP-96,486) antagonizes3H-LTD4 binding to guinea pig lung membranes and3H-PAF binding to rabbit platelets with Ki's of 20 and 24 nM respectively[1]. | ||
体内研究 (In Vivo) | CP-96486 (CP-96,486) inhibits iv LTD4- and iv PAF-induced bronchoconstriction in guinea pigs with ED50's of 0.27 and 0.26 mg/kg p.o. respectively[1]. | ||
分子量 | 502.99 | ||
Formula | C31H23ClN4O | ||
CAS 号 | 139401-45-9 | ||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |