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Neurokinin A(4-10)TFA
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Neurokinin A(4-10)TFA图片
包装与价格:
包装价格(元)
1mg电议
5mg电议
10mg电议
25mg电议
50mg电议
100mg电议

产品介绍
Neurokinin A (4-10) TFA 是速激肽NK2受体激动剂。
生物活性

Neurokinin A (4-10) TFA is atachykinin NK2receptoragonist[1].

IC50& Target

NK2receptor[1]

体外研究
(In Vitro)

Neurokinin A (NKA) and its truncated form NKA(4-10) are potent spasmogens of human colon circular muscle, an action mediated exclusively via tachykinin NK2receptors. A structure-activity study of the neurokinin A (NKA) fragment NKA(4-10) is performed to investigate the importance of amino acid residues for receptor efficacy, potency and affinity at the NK2receptor in human colon circular muscle. A high density of NK2receptors has been demonstrated in this tissue, using in vitro autoradiography and radioligand binding[1].

分子量

880.93

性状

Solid

Formula

C36H55F3N8O12S

Sequence

Asp-Ser-Phe-Val-Gly-Leu-Met-NH2

Sequence Shortening

DSFVGLM-NH2

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Sealed storage, away from moisture

Powder-80°C2 years
-20°C1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

溶解性数据
In Vitro: 

H2O :< 0.1 mg/mL(insoluble)