包装 | 价格(元) |
1mg | 电议 |
5mg | 电议 |
10mg | 电议 |
25mg | 电议 |
50mg | 电议 |
100mg | 电议 |
生物活性 | Neurokinin A (4-10) TFA is atachykinin NK2receptoragonist[1]. | ||||||
IC50& Target | NK2receptor[1] | ||||||
体外研究 (In Vitro) | Neurokinin A (NKA) and its truncated form NKA(4-10) are potent spasmogens of human colon circular muscle, an action mediated exclusively via tachykinin NK2receptors. A structure-activity study of the neurokinin A (NKA) fragment NKA(4-10) is performed to investigate the importance of amino acid residues for receptor efficacy, potency and affinity at the NK2receptor in human colon circular muscle. A high density of NK2receptors has been demonstrated in this tissue, using in vitro autoradiography and radioligand binding[1]. | ||||||
分子量 | 880.93 | ||||||
性状 | Solid | ||||||
Formula | C36H55F3N8O12S | ||||||
Sequence | Asp-Ser-Phe-Val-Gly-Leu-Met-NH2 | ||||||
Sequence Shortening | DSFVGLM-NH2 | ||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||
储存方式 | Sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) | ||||||
溶解性数据 | In Vitro: H2O :< 0.1 mg/mL(insoluble) |