OXA(17-33) TFA 是一种高效、选择性的orexin-1 receptor (OX1)激动剂。OXA(17-33) TFA 对 OX1 (EC50=8.29 nM) 的选择性比 OX2 (187 nM) 高 23 倍。
生物活性 | OXA(17-33) TFA is a potent and selectiveorexin-1 receptor (OX1)agonist. OXA(17-33) TFA shows a ~23-fold selectivity for the OX1 (EC50=8.29 nM) over OX2 (187 nM)[1]. |
IC50& Target | OX1 8.29 nM (EC50) | OX2 187 nM (EC50) |
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分子量 | |
Formula | |
Sequence | Tyr-Glu-Leu-Leu-His-Gly-Ala-Gly-Asn-His-Ala-Ala-Gly-Ile-Leu-Thr-Leu-NH2 |
Sequence Shortening | |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |