TCS-OX2-29 (hydrochloride) 是一种有效的,高亲和力和选择性的OX2R拮抗剂,其IC50值为 40 nM,pKI值为 7.5。与 OX1相比,TCS-OX2-29 对OX2的选择性约高了 250倍。
生物活性 | TCS-OX2-29 (hydrochloride) is a potent, high affinities and selectiveorexin-2 receptor (OX2R)antagonist with anIC50value of 40 nM and apKIvalue of 7.5. TCS-OX2-29 displays ~250-fold selectivity forOX2overOX1[1][2]. |
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运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |