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OT antagonist 1
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
OT antagonist 1图片
CAS NO:479080-38-1
包装与价格:
包装价格(元)
100mg电议
250mg电议
500mg电议

产品介绍
OT antagonist 1 (Compound 4) 是一种有效的选择性催产素 (Oxytocin) 拮抗剂,Ki为 50 nM。
生物活性

OT antagonist 1 (Compound 4) is a potent, selectiveOxytocinantagonist with aKiof 50 nM.

IC50& Target

Ki: 50 nM (Oxytocin)[1]

体外研究
(In Vitro)

Oxytocin (OT) is a nonapeptide hormone that acts on the OT receptor, a seven-transmembrane (7TM) (Gq-coupled) receptor. The OT receptor has no subtypes but is related to the vasopressin receptors V1A, V1Band V2. OT antagonists have therapeutic potential in a number of areas including pre-term labour: Benign Prostatic Hyperplasia and sexual dysfunction. As a result there is significant interest in the identification of potent, selective, orally bioavailable OT antagonists[1].

分子量

390.44

Formula

C22H22N4O3

CAS 号

479080-38-1

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.