CAS NO: | 500170-27-4 |
包装 | 价格(元) |
1mg | 电议 |
5mg | 电议 |
10mg | 电议 |
50mg | 电议 |
100mg | 电议 |
生物活性 | d[Cha4]-AVP is a potent and selectivevasopressin (AVP) V1b receptoragonist with aKiof 1.2 nM forhuman V1b receptor. d[Cha4]-AVP shows more selective for V1b receptor than human V1a receptor, V2 receptor, and oxytocin receptors[1][2]. | ||||||||||||||||
IC50& Target | Ki: 1.2 nM (vasopressin V1B receptor), 151 nM (vasopressin V1A receptor), 240 nM (Oxytocin receptor), 750 nM (vasopressin V2 receptor)[1] | ||||||||||||||||
体外研究 (In Vitro) | d[Cha4]-AVP binds to hV1b receptors and human oxytocin receptors with pKivalues of 9.68 and 7.68, respectively[2]. | ||||||||||||||||
分子量 | 1094.31 | ||||||||||||||||
性状 | Solid | ||||||||||||||||
Formula | C50H71N13O11S2 | ||||||||||||||||
CAS 号 | 500170-27-4 | ||||||||||||||||
Sequence | {Mpa}-Tyr-Phe-{Cha}-Asn-Cys-Pro-Arg-Gly-NH2 (Disulfide bridge:Mpa1-Cys6) | ||||||||||||||||
Sequence Shortening | {Mpa}YF{Cha}NCPRG-NH2 (Disulfide bridge:Mpa1-Cys6) | ||||||||||||||||
运输条件 | Room temperature in continental US; may vary elsewhere. | ||||||||||||||||
储存方式 | Sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) | ||||||||||||||||
溶解性数据 | In Vitro: H2O : 100 mg/mL(91.38 mM;Need ultrasonic) 配制储备液
* 请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |