Cutamesine (SA4503; AGY-94806) 是一种选择性sigma 1受体激动剂,IC50为 17.4 nM,而对 sigma 2 受体的亲和力低 100 倍。
生物活性 | Cutamesine (SA4503; AGY-94806) is a selective sigma 1 receptor(σ1R) agonist; high affinity for thesigma 1 receptorsubtype labeled by (+)-[3H]pentazocine (IC50= 17.4±1.9 nM); 100-fold less affinity for thesigma 2 receptor. |
Clinical Trial | |
分子量 | |
Formula | |
CAS 号 | |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |