GR 231118 是神经肽 Y C 末端的类似物,是一种有效的、竞争性的和相对选择性的人神经肽 Y Y 受体拮抗剂,pKi 为 10.4。
Cas No. | 158859-98-4 |
别名 | 1229U91; GW1229 |
化学名 | (6S,9Z,12Z,13Z,14aS,20S,23Z,26Z,27Z,28aS)-6,20-bis((Z)-((2S,3S)-2-amino-1-hydroxy-3-methylpentylidene)amino)-N'12,N'26-bis((6S,7Z,9S,10Z,12S,13Z,15S)-1-amino-12-(3-guanidinopropyl)-8,11,14-trihydroxy-6-((Z)-hydroxy(((S)-1-hydroxy-3-(4-hydroxyphenyl)-1-imi |
Canonical SMILES | CC[C@]([C@@](N)([H])/C(O)=N/[C@@](C1=O)([H])CC/C(O)=N/CC(/N=C(O)/[C@]2([H])CCCN2C([C@](/N=C(O)/[C@](N)([H])[C@@](CC)([H])C)([H])CC/C(O)=N/CC(/N=C(O)/[C@]3([H])CCCN31)([H])/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](/C(O)=N/[C@@](C(O)=N)([H])CC |
分子式 | C110H170N34O24 |
分子量 | 2352.77 |
溶解度 | Soluble in water |
储存条件 | Desiccate at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |