ROS 234 dioxalate 是一种有效的 H3 拮抗剂,对豚鼠回肠 H3 受体的 pKB 为 9.46,对大鼠大脑皮层 H3 受体的 pKi 为 8.90,在体外的 ED50 为 19.12 mg/kg (ip)大鼠大脑皮层。
Cas No. | 184576-87-2 |
化学名 | N-(3-(1H-imidazol-5-yl)propyl)-1H-benzo[d]imidazol-2-amine dioxalate |
Canonical SMILES | OC(C(O)=O)=O.OC(C(O)=O)=O.C1(CCCNC2=NC3=CC=CC=C3N2)=CN=CN1 |
分子式 | C13H15N5.2C2H2O4 |
分子量 | 421.37 |
溶解度 | <21.07mg/ml in Water;<21.07mg/ml in DMSO |
储存条件 | Desiccate at RT |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. |
Shipping Condition | Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |