CAS NO: | 1217623-85-2 |
包装 | 价格(元) |
1mg | 电议 |
10mg | 电议 |
25mg | 电议 |
生物活性 | Raclopride-d5 (hydrochloride) is the deuterium labeled Raclopride. Raclopride is adopamine D2/D3receptorantagonist, which binds toD2andD3receptors with dissociation constants (Kis) of 1.8 nM and 3.5 nM, respectively, but has a very low affinity for D1and D4receptors with Kis of 18000 nM and 2400 nM, respectively[1][2]. |
体外研究 (In Vitro) | Stable heavy isotopes of hydrogen, carbon, and other elements have been incorporated into drug molecules, largely as tracers for quantitation during the drug development process. Deuteration has gained attention because of its potential to affect the pharmacokinetic and metabolic profiles of drugs[1]. |
分子量 | 352.27 |
Formula | C15H16D5Cl3N2O3 |
CAS 号 | 1217623-85-2 |
中文名称 | 雷氯必利 d5 (盐酸盐) |
运输条件 | Room temperature in continental US; may vary elsewhere. |
储存方式 | Please store the product under the recommended conditions in the Certificate of Analysis. |