Thiocolchicoside 是秋水仙碱的半合成硫衍生物，是竞争性 GABAA 受体拮抗剂和甘氨酸受体拮抗剂。它是肌肉松弛剂，具有抗炎作用，可用于缓解疼痛的研究。

Thiocolchicoside (Muscoril, Myoril, Neoflax) is a muscle relaxant with anti-inflammatory and analgesic effects. It acts as a competitive GABAA receptor antagonist and also glycine receptor antagonist with similar potency and nicotinic acetylcholine receptors to a much lesser extent. It has powerful convulsant activity and should not be used in seizure-prone individuals.

602-41-5

C27H33NO10S

563.62

Thiocolchicine 2-glucoside analog;Coltramyl;硫秋水仙苷;硫秋水仙苷;噻可撒可

DMSO:177.4 mM
H2O:177.4 mM
Powder: -20°C for 3 years
In solvent: -80°C for 2 years