VU6015929 是一种活性双盘状结构域受体 1/2 (DDR1/2) 的抑制剂（IC50 分别为 4.67 nM 和 7.39 nM）。

VU6015929 is an inhibitor of active dual discoidin domain receptor 1/2 (DDR1/2)( IC50s of 4.67 nM and 7.39 nM, respectively).

VU6015929 potently blocks collagen-induced DDR1 activation and collagen-IV production, suggesting DDR1 inhibition as an exciting target for antifibrotic therapy[1].

2442597-56-8

C24H19F4N5O2

485.443

DMSO:250 mg/mL (515.01 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years