Edg-2 receptor inhibitor 1 是一种提取的 Edg-2 受体抑制剂 (IC50:<0.1 μM)。

Edg-2 receptor inhibitor 1 is an Edg-2 receptor inhibitor extracted (IC50:<0.1 μM).

Edg-2 receptor inhibitor 1 is an inhibitor of the endothelial differentiation gene receptor 2 (Edg-2, EDG2), which is activated by lysophosphatidic acid (LPA) and is also termed as LPA1 receptor, and is useful for the treatment of diseases such as atherosclerosis, myocardial infarction and heart failure, for example[1].

1195941-38-8

C27H27NO5

445.515

SAR-100842

DMSO:83.3 mg/mL (186.98 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years