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CB2 receptor agonist 2
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
CB2 receptor agonist 2图片
CAS NO:1314230-75-5
包装与价格:
包装价格(元)
1 mg电议
2 mg电议
5 mg电议
10 mg电议
25 mg电议
50 mg电议

产品名称
CB2受体拮抗剂2
ZINC72105556
4-Quinolone-3-Carboxamide Furan CB2 Agonist
产品介绍
CB2 receptor agonist 2 是有效和选择性的 CB2 受体激动剂。对 CB2 的 Ki 为 8.5 nM。CB2 receptor agonist 2 对 CB2 具有高亲和力和选择性。

产品描述

CB2 receptor agonist 2 is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor, Ki = 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2.

体外活性

CB2 receptor agonist 2 (compound 4g) (1 μM; 72 hours) shows low or no cytotoxicity to Hep-G2 cells[1].

体内活性

CB2 receptor agonist 2 (compound 4g) (1 and 3 mg/kg; 1 hour) is very potent (with maximal effect being reached already at the 1 mg/kg dose) and has antihyperalgesic effects, efficacious also on the first phase of the nocifensive response and strongly reduced by AM630, a CB2-selective antagonist/inverse agonist [1].

Cas No.

1314230-75-5

分子式

C30H36N2O4

分子量

488.62

别名

CB2受体拮抗剂2;ZINC72105556;4-Quinolone-3-Carboxamide Furan CB2 Agonist

储存和溶解度

DMSO:3mg/mL (6.1mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years