AKR1C3-IN-4 是醛酮还原酶 1C3 (AKR1C3) 选择性抑制剂，IC50为 0.56 μM。它在去势抵抗性前列腺癌中有研究的价值。

AKR1C3-IN-4 is a potent and selective inhibitor of aldo-keto reductase 1C3 (AKR1C3) with an IC50 of 0.56 μM. AKR1C3-IN-4 has the potential for castrate resistant prostate cancer (CRPC) research.

The IC50 of AKR1C3-IN-4 for AKR1C2 is 15.1 μM[1].

1284180-11-5

C14H10F3NO2

281.23

AKR1C3-IN-4

DMSO:100 mg/mL (355.58 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years