CCR1 antagonist 9 is an effective and selective CCR1 antagonist (IC50: 6.8 nM in calcium flux assay).

CCR1 antagonist 9 (Compound 19e) blocks the CCR1 chemotaxis of THP-1 cells (IC50: 28 nM) and also blocks hERG (IC50: 30 μM).

1220026-26-5

C20H16FN5O3S

425.44

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years