APY0201 是PIKfyve抑制剂，能够抑制 PtdIns3P 转化为PtdIns(3,5)P2 (IC50:5.2 nM)，还能够抑制IL-12/IL-23产生。

APY0201 is a effective, highly specific, ATP-competitive PIKfyve inhibitor (IC50: 5.2 nM). It can interrupt the conversion of phosphatidylinositol 3-phosphate (PtdIns3P) to PtdIns(3, 5)P2.

1232221-74-7

C23H23N7O

413.485

DMSO:~5 mg/mL (12.1 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years