AR-M 1000390 hydrochloride 是选择性 δ 阿片受体激动剂，EC50为 7.2±0.9 nM。

AR-M 1000390 (hydrochloride), also known as ARM-390, is a low-internalizing nonpeptidic δ-selective opioid receptor agonist; derivative of SNC 80. Does not trigger acute desensitization of the analgesic response; reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.

Does not trigger acute desensitization of the analgesic response

Reduces CFA-induced hyperalgesia. Brain penetrant following systemic administration.

209808-47-9

C23H29ClN2O

384.95

ARM390 Hydrochloride;ARM-390 HCl

H2O:38.49 mg/mL (100 mM)
DMSO:38.49 mg/mL (100 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years