Difelikefalin acetate 是一种外周受限的 kappa 阿片受体激动剂。CR845 表现出低 P450 CYP 抑制和对大脑的低渗透性。

Difelikefalin acetate is a peripherally restricted kappa opioid receptor agonist. CR845 exhibit low P450 CYP inhibition and low penetration into the brain.

TP2501

C38H57N7O8

739.9

Difelikefalin acetate(1024828-77-0 free base);CR 845 acetate;Difelikefalin醋酸盐;FE 202845 acetate

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years