BMS986187 是一种有效的δ-阿片受体选择性正变构调节剂 (PAM)，其EC50= 0.03 μM，pKB= 6.02 (~1 μM)。BMS986187 对 μ 受体无明显 PAM 活性 (EC50=3 μM)。

BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.

684238-37-7

C31H34O4

470.609

DMSO:10 mM
Powder: -20°C for 3 years
In solvent: -80°C for 2 years