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GSK9311
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
GSK9311图片
CAS NO:1923851-49-3
包装:100 mg
市场价:8247元

产品介绍

产品描述

GSK9311 inhibits BRPF bromodomain (pIC50: 6.0 and 4.3 for BRPF1 and BRPF2, respectively). GSK9311 is a less active analog of GSK6853. It can be used as a negative control.

体外活性

GSK6853 is a less active analogue of GSK6853 in which the 5-amide is alkylated. GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain. GSK6853 shows properties suitable for cellular and in vivo studies[1].

Cas No.

1923851-49-3

分子式

C24H31N5O3

分子量

437.53

储存和溶解度

DMSO:30 mg/mL (68.57 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years