Enzalutamide carboxylic acid 是 Enzalutamide 非活性代谢物。Enzalutamide 是雄激素受体 (AR) 拮抗剂。

Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .

Enzalutamide is an oral agent for the treatment of metastatic castration-resistant prostate cancer (mCRPC);?N-desmethyl enzalutamide is its active metabolite, which has clinically relevant anti-androgen capacities similar to enzalutamide, and carboxylic acid enzalutamide is an inactive metabolite.

1242137-15-0

C20H13F4N3O3S

451.4

DMSO:10 mM
Powder: -20°C for 3 years
In solvent: -80°C for 2 years