2-hydroxy Flutamide 是 Flutamide 的活性代谢物，是雄激素受体拮抗剂，其IC50值为700 nM。它可用于研究前列腺癌。

2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancer

The pharmacologically active metabolite 2-hydroxy-flutamide, this principle metabolite increased CYP3A metabolism of midazolam in human microsomes (30%) and hepatocytes (110%)[1].

52806-53-8

C11H11F3N2O4

292.214

DMSO:25mg/ml(85.5 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years