NF-56-EJ40 是一种有效且高度特异性的人 SUCNR1 拮抗剂,IC50 为 25 nM,Ki 为 33 nM。
产品描述
NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of 25 nM and a Ki of 33 nM.
体外活性
NF-56-EJ40 shows a high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM. NF-56-EJ40 shows almost no activity towards rat SUCNR1[1].
Cas No.
2380230-73-7
分子式
C27H29N3O3
分子量
443.54
储存和溶解度
H2O:4.55 mg/mL (10.26 mM),ultrasonic and adjust pH to 9 with NaOH
DMSO:5 mg/mL (11.27 mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years