GLP-1R Antagonist 1 (compound 5d) 是口服有效的、能透过中枢神经系统的，胰高血糖素样肽 1 受体 (GLP-1R) 的非竞争性抑制，其IC50 值为 650 nM。

GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).

488097-06-9

C16H11ClF6N4O2

440.73

DMSO:90mg/mL (204.2mM),Need ultrasonic
Powder: -20°C for 3 years
In solvent: -80°C for 2 years