Selective PAR2 peptide antagonist. Reverses taxol-induced mechanical allodynia, heat hyperalgesia and PKC activation in ICR mice. Blocks ERK activation and collagen production in isolated cardiac fibroblasts. Also reduces symptoms in a mouse model of dermatophyte-associated itch.

245329-02-6

C39H60N10O8

796.97

H2O:1 mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years