GAK inhibitor 49 是 ATP 竞争性的细胞周期蛋白G相关激酶选择性抑制剂，Ki=0.54 nM，细胞IC50=56 nM。它也具有与 RIPK2 结合的能力。

GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).

319492-82-5

C20H22N2O5

370.405

DMSO:10 mM
Powder: -20°C for 3 years
In solvent: -80°C for 2 years