CARM1-IN-1 shows high and selective CARM1 inhibition, with lower or no activity against a panel of different PRMTs or HKMTs. In human LNCaP cells, CARM1-IN-1 dose-dependently reduces of the PSA promoter activity.

T10682

C26H22Br2ClNO3

591.72

CARM1-IN-1 hydrochloride

DMSO:38 mg/mL (64.22 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years