HA155 是一种高效的 ATX 选择性抑制剂，其IC50=5.7 nM。

HA155 selectively and potently inhibits autotaxin with an IC50 of 5.7 nM.

HA155 completely attenuates the thrombin-mediated increase in platelet-derived LPA dose-dependently [2].HA155 is an ATX inhibitor by binding to the ATX active site [3].

1312201-00-5

C24H19BFNO5S

463.29

CS-963

DMSO:8 mg/mL (17.27 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years