Mu Opioid Receptor antagonist 3 (compound 26) 是一种有效且具有选择性的μ 阿片受体 (MOR)拮抗剂，Ki为 0.24 nM，EC50为 0.54 nM。Mu Opioid Receptor antagonist 3 对吗啡具有显著的中枢神经系统拮抗作用，与 Naloxone 相比，其诱发戒断症状较少。Mu Opioid Receptor antagonist 3 可用于阿片类药物使用障碍 (OUD) 的研究。

Mu opioid receptor antagonist 3 (compound 26) is a potent and selective μ opioid receptor (MOR) antagonist with a K i of 0.24 nM and an EC 50 of 0.54 nM. Mu opioid receptor antagonist 3 has remarkable CNS antagonism against morphine, and precipitated fewer withdrawal symptoms than Naloxone. Mu opioid receptor antagonist 3 can be used for researching opioid use disorders (OUD) [1].

C25H28N2O4S

452.57

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years