GSK-5498A is a selective blocker of CARC (IC50, 1 μM). It inhibits mediator release from mast cells, and pro-inflammatory cytokine release from T-cells in a variety of species.

1253186-49-0

C18H11F6N3O

399.29

GSK-5498A

DMSO:100 mg/mL (250.44 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years