TC-DAPK 6 is an effective, ATP-competitive, and highly selective inhibitor of DAPK (IC50=69 and 225 nM against DAPK1 and DAPK3, respectively, with 10 μM ATP).

TC-DAPK 6 is found to be the most potent Death-associated protein kinase inhibitor with enzyme selectivity. TC-DAPK 6 also inhibits p70S6K (1 μM< IC50< 10 μM)[1].

315694-89-4

C17H12N2O2

276.29

TC-DAPK 6

DMSO:18.67 mg/mL (67.57 mM),Need ultrasonic and warming
Powder: -20°C for 3 years
In solvent: -80°C for 2 years