GCN2-IN-1 是一种有效的一般性调控阻遏蛋白激酶 2 抑制剂,可作为化疗药物用于癌症治疗的研究。
产品描述
GCN2-IN-1 is an effective GCN2 inhibitor and can be used in research on the treatment of cancer as a chemotherapeutic agent.
体外活性
GCN2-IN-1 inhibits GCN2 with an IC50 of<0.3 μM in the enzyme assay and an IC50 of 0.3-3 μM in the cell assay[1].
Cas No.
1448693-69-3
分子式
C19H18N10O
分子量
402.41
别名
A-92;GCN2-IN-1
储存和溶解度
DMSO:55mg/mL (136.68 mM),Need ultrasonic and warming
Powder: -20°C for 3 years
In solvent: -80°C for 2 years