产品描述
CDD0102 is a potent agonist of M1 Muscarinic receptor.
体外活性
CDD0102 displays much lower activity at M3 and M5 receptors.
体内活性
CDD0102 (i.p.) crosses the blood-brain barrier (BBB) in a dose-dependent manner. In toxicological studies, the LD50 of CDD0102 is 190 mg/kg following i.p. injections and greater than 1,000 mg/kg following oral administration. CDD0102 (10 mg/kg) fully reverses memory deficits associated with IgG-192 saporin administration. Again, no side effects are observed at this dose.
Cas No.
146422-58-4
分子式
C8H12N4O
分子量
180.21
别名
CDD0102A;CDD0102
储存和溶解度
(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years