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KT109
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
KT109图片
CAS NO:1402612-55-8
包装:5 mg
市场价:7000元

产品名称
KT-109
KT 109
产品介绍

产品描述

KT109 is a selective inhibitor of DAGLβ (IC50 = 42 nM). KT109-treated wild-type mice displayed reductions in LPS-induced allodyni as well as in DAGL-β (-/-) micea. Repeated KT109 administration prevented the expression of LPS-induced allodynia, without evidence of tolerance. Intraplantar injection of KT109 into the LPS-treated paw, but not the contralateral paw, reversed the allodynic responses. KT109 also reversed allodynia in the CCI and CINP models and lacked discernible side effects (e.g. anxiogenic behaviour, gross motor deficits or gastric ulcers).

Cas No.

1402612-55-8

分子式

C27H26N4O

分子量

422.52

别名

KT-109;KT 109;KT109

储存和溶解度

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years