Selective TRPC5 activator (EC50 = 1.4 μM in a calcium influx assay, 1.3 μM in whole cell patch clamp assay). Displays >14.5-fold selectivity for TRPC5 over other TRP channels (EC50 = 20.6 μM for TRPM8). Also activates TRPC1:5 and TRPC4:5 heteromers.

896684-04-1

C24H33N3O4S

459.61

BTD

DMSO:Soluble
Powder: -20°C for 3 years
In solvent: -80°C for 2 years