UNC0379 TFA 是一个选择性的底物竞争性的赖氨酸甲基转移酶SETD8(KMT5A) 抑制剂，IC50值为 7.3 μM，对其他 15 种甲基转移酶有很好的选择性。

UNC0379 TFA is a selective, substrate-competitive inhibitor of lysine methyltransferase SETD8 ( KMT5A ) with an IC 50 of 7.3 μM; selective over 15 other methyltransferases [1].

1620401-83-3

C25H36F3N5O4

527.589

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years