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ZK824859 hydrochloride(2271122-53-1 free base)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
ZK824859 hydrochloride(2271122-53-1 free base)图片
包装与价格:
包装价格(元)
5 mg电议
10 mg电议
50 mg电议
100 mg电议
200 mg电议
500 mg电议
1 mL*10 mM(in DMSO)电议

产品名称
ZK824859 hydrochloride
ZK824859 hydrochloride (2271122-53-1 free base)
产品介绍

产品描述

ZK824859 hydrochloride is an oral available and selective inhibitor of urokinase plasminogen activator (uPA)(IC50s of 79 nM, 1580 nM and 1330 nM for human uPA, tPA, and plasmin, respectively).

体外活性

ZK824859 is 5 fold less potent and has lost selectivity in mouse: uPA with IC50 of 410?nM; tPA with IC50 of 910?nM; plasmin with IC50 of 1600?nM compared to human IC50 of 79?nM, 1580?nM and 1330?nM respectively.

Cas No.

T13409L

分子式

C23H23ClF2N2O4

分子量

464.89

别名

ZK824859 hydrochloride;ZK824859 hydrochloride (2271122-53-1 free base)

储存和溶解度

DMSO:125 mg/mL (268.88 mM)
Powder: -20°C for 3 years
In solvent: -80°C for 2 years