GSK1820795A 作为替米沙坦类似物是hGPR132a的选择性拮抗剂。GSK1820795A阻断了 N-acylamides 对表达hGPR132a的酵母细胞的活化。

GSK1820795A, as a telmisartan analog, is a selective hGPR132a antagonist. GSK1820795A blocks activation of yeast cells expressing hGPR132a by N-acylamides [1].

GSK1820795A blocks responses of yeast expressing hGPR132a to agonists NPGly, NLGly, linoleamide, and SB-583831 [1].

C35H34N8

566.7

(< 1 mg/ml refers to the product slightly soluble or insoluble )
Powder: -20°C for 3 years
In solvent: -80°C for 2 years