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BMY-14802 hydrochloride
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
BMY-14802 hydrochloride图片
CAS NO:105565-55-7
包装:5 mg
市场价:7000元

产品名称
BMY 14802 hydrochloride
产品介绍

产品描述

The theoretical role of sigma receptors in psychosis has led to the discovery of selective sigma receptor ligands as potential antipsychotic agents. BMY 14802 is a sigma receptor ligand (IC50: 112 nM for (+)-[3H]-3-PPP).

体外活性

In vitro: BMY 14802 has its most potent binding at the sigma binding site, with some degree of serotonin subtype 1A and negligible dopamine receptor binding [1].

体内活性

In vivo: BMY 14802 is atypical of standard neuroleptics in that it does not induce catalepsy in rats. In addition, it has been shown to have efficacy in animal models of psychosis [1].

Cas No.

105565-55-7

分子式

C18H23ClF2N4O

分子量

384.85

别名

BMY 14802 hydrochloride;BMY-14802 hydrochloride

储存和溶解度

H2O:<9.62mg/ml
Powder: -20°C for 3 years
In solvent: -80°C for 2 years