Potent, metabolically stable neurotensin receptor agonist peptide (IC50 = 0.15 nM for inhibition of [125I]-NT binding to neonatal mouse brain; EC50 = 1.9 nM for contraction of guinea pig ileum). Produces long-lasting hypothermic, neuroprotective and analgesic effects in mice following central administration in vivo.

139026-66-7

C38H66N8O7

746.96

JMV 449

H2O:0.80 mg/mL
Powder: -20°C for 3 years
In solvent: -80°C for 2 years