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Bitopertin(RG-1678 RO-4917838)
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验。
Bitopertin(RG-1678 RO-4917838)图片
CAS NO:845614-11-1
规格:≥98%
包装与价格:
包装价格(元)
5mg电议
10mg电议
25mg电议
50mg电议
100mg电议
250mg电议
500mg电议

产品介绍

Bitopertin (Paliflutine; RG1678; RO4917838; RG-1678; RO-4917838) is a novel, potent and non-competitive glycine reuptake inhibitor that inhibits human GlyT1 with an IC50 of 25 nM. GlyT1 is a key membrane transporter required to supply developing red blood cells with sufficient glycine to support erythropoiesis. It is under development as an adjunct to antipsychotics for the treatment of persistent negative symptoms or suboptimally-controlled positive symptoms associated with schizophrenia. Bitopertin-mediated glycine reuptake inhibition may represent a novel treatment option for schizophrenia, with the potential to address negative symptoms.

纯度:≥98%

CAS:845614-11-1