BD1008 is a selective antagonist of the sigma 1 (σ1) receptor (Ki = 2 nM) that exhibits 4-fold selectivity for σ1 over σ2. BD-1008 attenuate the toxicity and stimulant effects of cocaine through antagonism of sigma receptors References: Matsumoto RR, Gilmore DL, Pouw B, Bowen WD, Williams W, Kausar A, Coop A. Novel analogs of the sigma receptor ligand BD1008 attenuate cocaine-induced toxicity in mice. Eur J Pharmacol. 2004 May 10;492(1):21-6. PubMed PMID: 15145701.

纯度：≥98%

CAS：138356-09-9