CP-809101 (CP809101) is a selective 5-HT2C
receptor agonist with antipsychotic activity. It activates human
5-HT2C/5-HT2B/5-HT2A receptors with pEC50 of 9.96/7.19/6.81,
respectively. CP-809101 reduces motor impulsivity and reinstatement of
food seeking behavior in male rats. CP-809101 (0.3-3 mg/kg SC) reduced
responding for both nicotine and food and blocked the discriminative
stimulus properties of nicotine in a similar manner to lorcaserin and Ro
60-0175.
纯度:≥98%
CAS:479683-64-2